Shaffer, Christopher L

The discovery and characterization of the α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor potentiator N-propane-2-sulfonamide (PF-04958242). [electronic resource] - Journal of medicinal chemistry May 2015 - 4291-308 p. digital

Publication Type: Journal Article

1520-4804

10.1021/acs.jmedchem.5b00300 doi


Administration, Oral
Adolescent
Adult
Aged
Animals
Binding Sites
Disease Models, Animal
Dogs
Dose-Response Relationship, Drug
Drug Discovery
Drug Evaluation, Preclinical--methods
Drug Stability
Female
Humans
Male
Memory, Short-Term--drug effects
Mice, Inbred C57BL
Middle Aged
Protein Conformation
Rats, Sprague-Dawley
Receptors, AMPA--metabolism
Schizophrenia--drug therapy
Structure-Activity Relationship
Sulfonamides--chemistry
Thiophenes--chemistry
Young Adult