Mukerjee, Anindita

A nanotherapy strategy significantly enhances anticryptosporidial activity of an inhibitor of bifunctional thymidylate synthase-dihydrofolate reductase from Cryptosporidium. [electronic resource] - Bioorganic & medicinal chemistry letters 2015 - 2065-7 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1464-3405

10.1016/j.bmcl.2015.03.091 doi


Antiprotozoal Agents--chemical synthesis
Binding Sites
Cells, Cultured
Cryptosporidium--drug effects
Drug Synergism
Models, Molecular
Multienzyme Complexes--antagonists & inhibitors
Nanoparticles--chemistry
Tetrahydrofolate Dehydrogenase
Thymidylate Synthase--antagonists & inhibitors