Toward Labeled Argininamide-Type NPY Y1 Receptor Antagonists: Identification of a Favorable Propionylation Site in BIBO3304. [electronic resource]
- Archiv der Pharmazie Jun 2015
- 390-8 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
1521-4184
10.1002/ardp.201400427 doi
Animals Arginine--analogs & derivatives Binding Sites Binding, Competitive CHO Cells Cricetulus Dose-Response Relationship, Drug Drug Design Ligands Molecular Structure Propionates--chemical synthesis Protein Binding Radioligand Assay Receptors, Neuropeptide Y--antagonists & inhibitors Structure-Activity Relationship Transfection