Inhibition of Lapatinib-Induced Kinome Reprogramming in ERBB2-Positive Breast Cancer by Targeting BET Family Bromodomains. [electronic resource]
- Cell reports Apr 2015
- 390-404 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
2211-1247
10.1016/j.celrep.2015.03.037 doi
Antineoplastic Agents--pharmacology Blotting, Western Breast Neoplasms--metabolism Cell Line, Tumor Drug Resistance, Neoplasm--physiology Female Humans Lapatinib Mass Spectrometry Oligonucleotide Array Sequence Analysis Polymerase Chain Reaction Protein Kinase Inhibitors--pharmacology Proteomics Quinazolines--pharmacology Receptor, ErbB-2--metabolism Signal Transduction--physiology Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization