TY - GEN AU - Theodoulou,Natalie H AU - Bamborough,Paul AU - Bannister,Andrew J AU - Becher,Isabelle AU - Bit,Rino A AU - Che,Ka Hing AU - Chung,Chun-wa AU - Dittmann,Antje AU - Drewes,Gerard AU - Drewry,David H AU - Gordon,Laurie AU - Grandi,Paola AU - Leveridge,Melanie AU - Lindon,Matthew AU - Michon,Anne-Marie AU - Molnar,Judit AU - Robson,Samuel C AU - Tomkinson,Nicholas C O AU - Kouzarides,Tony AU - Prinjha,Rab K AU - Humphreys,Philip G TI - Discovery of I-BRD9, a Selective Cell Active Chemical Probe for Bromodomain Containing Protein 9 Inhibition SN - 1520-4804 PY - 2016///0726 KW - Amino Acid Sequence KW - Binding Sites KW - Cell Line KW - Crystallography, X-Ray KW - Drug Discovery KW - Humans KW - Models, Molecular KW - Molecular Docking Simulation KW - Small Molecule Libraries KW - chemistry KW - Transcription Factors KW - antagonists & inhibitors N1 - Publication Type: Journal Article; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1021/acs.jmedchem.5b00256 ER -