Oda, Shingo

Targeted screen for human UDP-glucuronosyltransferases inhibitors and the evaluation of potential drug-drug interactions with zafirlukast. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals Jun 2015 - 812-8 p. digital

Publication Type: Journal Article

1521-009X

10.1124/dmd.114.062141 doi


Drug Evaluation, Preclinical
Drug Interactions
Enzyme Inhibitors--adverse effects
Glucuronosyltransferase--antagonists & inhibitors
Humans
Indoles
Intestinal Mucosa--drug effects
Intestine, Small--drug effects
Isoenzymes--antagonists & inhibitors
Kinetics
Leukotriene Antagonists--adverse effects
Metabolic Detoxication, Phase II
Microsomes--drug effects
Microsomes, Liver--drug effects
Phenylcarbamates
Raloxifene Hydrochloride--metabolism
Recombinant Proteins--chemistry
Selective Estrogen Receptor Modulators--metabolism
Small Molecule Libraries
Substrate Specificity
Sulfonamides
Tosyl Compounds--adverse effects