Yang, Li

In vitro and in vivo efficacy of a potent opioid receptor agonist, biphalin, compared to subtype-selective opioid receptor agonists for stroke treatment. [electronic resource] - Brain research Jun 2015 - 1-11 p. digital

Publication Type: Comparative Study; Journal Article; Research Support, N.I.H., Extramural

1872-6240

10.1016/j.brainres.2015.03.022 doi


3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer--chemistry
Analgesics, Opioid--chemistry
Brain Edema--drug therapy
Brain Infarction--drug therapy
Brain Ischemia--drug therapy
Cells, Cultured
Enkephalin, Ala(2)-MePhe(4)-Gly(5)---chemistry
Enkephalin, D-Penicillamine (2,5)---chemistry
Enkephalins--chemistry
Glutamic Acid--toxicity
Ischemia--drug therapy
Motor Activity--drug effects
Neurons--drug effects
Neuroprotective Agents--chemistry
Receptors, Opioid, delta--agonists
Receptors, Opioid, kappa--agonists
Receptors, Opioid, mu--agonists
Reperfusion Injury--drug therapy
Severity of Illness Index
Stroke--drug therapy