Cohen, Anita

Discovery of new thienopyrimidinone derivatives displaying antimalarial properties toward both erythrocytic and hepatic stages of Plasmodium. [electronic resource] - European journal of medicinal chemistry May 2015 - 16-28 p. digital

Publication Type: Journal Article

1768-3254

10.1016/j.ejmech.2015.03.011 doi


Animals
Antimalarials--chemistry
CHO Cells
Cell Proliferation--drug effects
Cricetinae
Cricetulus
Drug Discovery
Erythrocytes--drug effects
Hep G2 Cells
Humans
Liver--drug effects
Malaria--drug therapy
Male
Mice
Parasitemia--drug therapy
Plasmodium falciparum--drug effects
Pyrimidines--chemistry
Structure-Activity Relationship
Trophozoites--drug effects