Discovery of new thienopyrimidinone derivatives displaying antimalarial properties toward both erythrocytic and hepatic stages of Plasmodium. [electronic resource]
- European journal of medicinal chemistry May 2015
- 16-28 p. digital
Publication Type: Journal Article
1768-3254
10.1016/j.ejmech.2015.03.011 doi
Animals Antimalarials--chemistry CHO Cells Cell Proliferation--drug effects Cricetinae Cricetulus Drug Discovery Erythrocytes--drug effects Hep G2 Cells Humans Liver--drug effects Malaria--drug therapy Male Mice Parasitemia--drug therapy Plasmodium falciparum--drug effects Pyrimidines--chemistry Structure-Activity Relationship Trophozoites--drug effects