Liu, Yong

The Discovery of Orally Bioavailable Tyrosine Threonine Kinase (TTK) Inhibitors: 3-(4-(heterocyclyl)phenyl)-1H-indazole-5-carboxamides as Anticancer Agents. [electronic resource] - Journal of medicinal chemistry Apr 2015 - 3366-92 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.

1520-4804

10.1021/jm501740a doi


Administration, Oral
Animals
Cell Cycle Proteins--antagonists & inhibitors
Cell Line, Tumor
Colon--drug effects
Colonic Neoplasms--drug therapy
Crystallography, X-Ray
Female
Humans
Indazoles--administration & dosage
Mice, Nude
Models, Molecular
Protein Kinase Inhibitors--administration & dosage
Protein Serine-Threonine Kinases--antagonists & inhibitors
Protein-Tyrosine Kinases--antagonists & inhibitors