Triapine-mediated ABCB1 induction via PKC induces widespread therapy unresponsiveness but is not underlying acquired triapine resistance. [electronic resource]
- Cancer letters May 2015
- 112-20 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1872-7980
10.1016/j.canlet.2015.02.049 doi
ATP Binding Cassette Transporter, Subfamily B--genetics Antineoplastic Agents--pharmacology Apoptosis--drug effects Blotting, Western Cell Proliferation--drug effects Colorectal Neoplasms--drug therapy Comparative Genomic Hybridization DNA Methylation--drug effects Drug Resistance, Multiple--drug effects Drug Resistance, Neoplasm--drug effects Humans Promoter Regions, Genetic--genetics Protein Kinase C--antagonists & inhibitors Pyridines--pharmacology RNA, Messenger--genetics RNA, Small Interfering--pharmacology Real-Time Polymerase Chain Reaction Reverse Transcriptase Polymerase Chain Reaction Thiosemicarbazones--pharmacology Tumor Cells, Cultured