Perturbation of the c-Myc-Max protein-protein interaction via synthetic α-helix mimetics. [electronic resource]
- Journal of medicinal chemistry Apr 2015
- 3002-24 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1520-4804
10.1021/jm501440q doi
Antineoplastic Agents--chemistry Basic Helix-Loop-Helix Leucine Zipper Transcription Factors--chemistry Cell Cycle Checkpoints--drug effects Cell Line, Tumor--drug effects Cell Proliferation--drug effects Chemistry Techniques, Synthetic Dose-Response Relationship, Drug Drug Design Drug Evaluation, Preclinical--methods Electrophoretic Mobility Shift Assay Helix-Loop-Helix Motifs Humans Inhibitory Concentration 50 Molecular Mimicry Nuclear Magnetic Resonance, Biomolecular Protein Multimerization Proto-Oncogene Proteins c-myc--antagonists & inhibitors Small Molecule Libraries--chemistry Surface Plasmon Resonance