Jung, Kwan-Young

Perturbation of the c-Myc-Max protein-protein interaction via synthetic α-helix mimetics. [electronic resource] - Journal of medicinal chemistry Apr 2015 - 3002-24 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1520-4804

10.1021/jm501440q doi


Antineoplastic Agents--chemistry
Basic Helix-Loop-Helix Leucine Zipper Transcription Factors--chemistry
Cell Cycle Checkpoints--drug effects
Cell Line, Tumor--drug effects
Cell Proliferation--drug effects
Chemistry Techniques, Synthetic
Dose-Response Relationship, Drug
Drug Design
Drug Evaluation, Preclinical--methods
Electrophoretic Mobility Shift Assay
Helix-Loop-Helix Motifs
Humans
Inhibitory Concentration 50
Molecular Mimicry
Nuclear Magnetic Resonance, Biomolecular
Protein Multimerization
Proto-Oncogene Proteins c-myc--antagonists & inhibitors
Small Molecule Libraries--chemistry
Surface Plasmon Resonance