Yhhu981, a novel compound, stimulates fatty acid oxidation via the activation of AMPK and ameliorates lipid metabolism disorder in ob/ob mice. [electronic resource]
- Acta pharmacologica Sinica Mar 2015
- 343-52 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1745-7254
10.1038/aps.2014.147 doi
AMP-Activated Protein Kinases--antagonists & inhibitors Acetyl-CoA Carboxylase--metabolism Alkynes--pharmacology Animals Anti-Obesity Agents--pharmacology Disease Models, Animal Dose-Response Relationship, Drug Energy Metabolism--drug effects Enzyme Activation Enzyme Activators--pharmacology Fatty Acids--metabolism Hep G2 Cells Humans Liver--drug effects Mice, Obese Muscle Fibers, Skeletal--drug effects Obesity--drug therapy Oxidation-Reduction Phosphorylation Protein Kinase Inhibitors--pharmacology Resorcinols--pharmacology Signal Transduction--drug effects Up-Regulation