Nirogi, Ramakrishna

Evaluation of metabolism dependent inhibition of CYP2B6 mediated bupropion hydroxylation in human liver microsomes by monoamine oxidase inhibitors and prediction of potential as perpetrators of drug interaction. [electronic resource] - Chemico-biological interactions Mar 2015 - 9-20 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1872-7786

10.1016/j.cbi.2015.01.028 doi


Bupropion--metabolism
Clorgyline--pharmacology
Cytochrome P-450 CYP2B6--metabolism
Cytochrome P-450 CYP2B6 Inhibitors--pharmacology
Drug Interactions
Glutathione--metabolism
Humans
Hydroxylation
Inhibitory Concentration 50
Kinesics
Microsomes, Liver--drug effects
Monoamine Oxidase Inhibitors--chemistry
Pargyline--pharmacology
Phenelzine--pharmacology
Selegiline--pharmacology