Price, Kerry L Varenicline Interactions at the 5-HT3 Receptor Ligand Binding Site are Revealed by 5-HTBP. [electronic resource] - ACS chemical neuroscience Jul 2015 - 1151-7 p. digital Publication Type: Journal Article; Research Support, Non-U.S. Gov't ISSN: 1948-7193 Standard No.: 10.1021/cn500369h doi Subjects--Topical Terms: Amino Acid SequenceAnimalsBinding Sites--drug effectsCarrier Proteins--geneticsCrystallography, X-RayHEK293 CellsHumansHydrogen BondingMiceModels, MolecularMutationOocytesPatch-Clamp TechniquesProtein Structure, SecondaryReceptors, Serotonin, 5-HT3--geneticsSerotonin--metabolismSerotonin Agents--metabolismVarenicline--metabolismWater--metabolismXenopus