Ishchenko, Alexey

Structure-based design of low-nanomolar PIM kinase inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Feb 2015 - 474-80 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2014.12.041 doi


Binding Sites
Crystallography, X-Ray
Drug Design
Hydrogen Bonding
Molecular Dynamics Simulation
Protein Binding
Protein Isoforms--antagonists & inhibitors
Protein Kinase Inhibitors--chemical synthesis
Protein Structure, Tertiary
Proto-Oncogene Proteins c-pim-1--antagonists & inhibitors
Static Electricity
Structure-Activity Relationship