Brand, Michael

Small molecule inhibitors of bromodomain-acetyl-lysine interactions. [electronic resource] - ACS chemical biology Jan 2015 - 22-39 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Review

1554-8937

10.1021/cb500996u doi


Acetylation
Animals
Histones--metabolism
Humans
Ligands
Lysine--metabolism
Models, Molecular
Nuclear Proteins--antagonists & inhibitors
Protein Binding
Protein Processing, Post-Translational--drug effects
Protein Structure, Tertiary
Small Molecule Libraries--chemistry
Structure-Activity Relationship