Ivanenkov, Yan A

Design, synthesis and biological evaluation of novel potent MDM2/p53 small-molecule inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Jan 2015 - 404-9 p. digital

Publication Type: Evaluation Study; Journal Article; Research Support, Non-U.S. Gov't

1464-3405

10.1016/j.bmcl.2014.09.070 doi


Antineoplastic Agents--chemical synthesis
Cell Proliferation--drug effects
Drug Design
Humans
Models, Molecular
Molecular Dynamics Simulation
Molecular Structure
Neoplasms--drug therapy
Proto-Oncogene Proteins c-mdm2--antagonists & inhibitors
Small Molecule Libraries--chemical synthesis
Structure-Activity Relationship
Tumor Cells, Cultured
Tumor Suppressor Protein p53--antagonists & inhibitors