Tariquidar inhibits P-glycoprotein drug efflux but activates ATPase activity by blocking transition to an open conformation. [electronic resource]
- Biochemical pharmacology Dec 2014
- 558-66 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1873-2968
10.1016/j.bcp.2014.10.006 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors Adenosine Triphosphatases--chemistry Animals Cell Line Cricetinae Drug Resistance, Multiple Protein Conformation Quinolines--pharmacokinetics