TY - GEN AU - Cohrs,Björn AU - Zhao,Yi AU - Lützen,Ulf AU - Culman,Juraj AU - Clement,Bernd AU - Zuhayra,Maaz TI - In vivo SPECT imaging of [¹²³I]-labeled pentamidine pro-drugs for the treatment of human African trypanosomiasis, pharmacokinetics, and bioavailability studies in rats SN - 1873-3476 PY - 2016///0321 KW - Administration, Oral KW - Animals KW - Biological Availability KW - Blood-Brain Barrier KW - metabolism KW - Brain KW - Humans KW - Male KW - Pentamidine KW - analogs & derivatives KW - Prodrugs KW - Rats KW - Rats, Sprague-Dawley KW - Succinates KW - pharmacokinetics KW - Time Factors KW - Tissue Distribution KW - Tomography, Emission-Computed, Single-Photon KW - methods KW - Trypanocidal Agents KW - Trypanosomiasis, African KW - drug therapy N1 - Publication Type: Comparative Study; Journal Article UR - https://doi.org/10.1016/j.ijpharm.2014.10.032 ER -