Cohrs, Björn

In vivo SPECT imaging of [¹²³I]-labeled pentamidine pro-drugs for the treatment of human African trypanosomiasis, pharmacokinetics, and bioavailability studies in rats. [electronic resource] - International journal of pharmaceutics Dec 2014 - 167-75 p. digital

Publication Type: Comparative Study; Journal Article

1873-3476

10.1016/j.ijpharm.2014.10.032 doi


Administration, Oral
Animals
Biological Availability
Blood-Brain Barrier--metabolism
Brain--metabolism
Humans
Male
Pentamidine--analogs & derivatives
Prodrugs
Rats
Rats, Sprague-Dawley
Succinates--pharmacokinetics
Time Factors
Tissue Distribution
Tomography, Emission-Computed, Single-Photon--methods
Trypanocidal Agents--pharmacokinetics
Trypanosomiasis, African--drug therapy