Yan, Chao

Discovery and characterization of small molecules that target the GTPase Ral. [electronic resource] - Nature Nov 2014 - 443-7 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1476-4687

10.1038/nature13713 doi


ATP-Binding Cassette Transporters--metabolism
Animals
Cell Line, Tumor
Cell Proliferation--drug effects
Computer Simulation
Drug Screening Assays, Antitumor
Female
GTPase-Activating Proteins--metabolism
Humans
Mice
Models, Molecular
Molecular Targeted Therapy
Neoplasms--drug therapy
Protein Binding--drug effects
Signal Transduction--drug effects
Small Molecule Libraries--chemistry
Substrate Specificity
Xenograft Model Antitumor Assays
ral GTP-Binding Proteins--antagonists & inhibitors
ras Proteins--metabolism