Srinivasrao, Ganipisetti

Design and synthesis of a cell-permeable, drug-like small molecule inhibitor targeting the polo-box domain of polo-like kinase 1. [electronic resource] - PloS one 2014 - e107432 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1932-6203

10.1371/journal.pone.0107432 doi


Antineoplastic Agents--chemical synthesis
Benzimidazoles--chemical synthesis
Catalytic Domain
Cell Cycle Proteins--antagonists & inhibitors
Cell Membrane Permeability
Drug Design
Drug Screening Assays, Antitumor
HeLa Cells
Humans
Models, Molecular
Organophosphates--chemical synthesis
Protein Binding
Protein Kinase Inhibitors--chemical synthesis
Protein Serine-Threonine Kinases--antagonists & inhibitors
Proto-Oncogene Proteins--antagonists & inhibitors
Polo-Like Kinase 1