Asamitsu, Sefan
Sequence-specific DNA alkylation and transcriptional inhibition by long-chain hairpin pyrrole-imidazole polyamide-chlorambucil conjugates targeting CAG/CTG trinucleotide repeats. [electronic resource]
- Bioorganic & medicinal chemistry Sep 2014
- 4646-57 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3391
10.1016/j.bmc.2014.07.019 doi
Alkylation--drug effects
Chlorambucil--chemistry
DNA--drug effects
Imidazoles--chemistry
Nylons--chemistry
Pyrroles--chemistry
Structure-Activity Relationship
Transcription, Genetic--drug effects
Trinucleotide Repeats--drug effects