TY  - GEN
AU  - Bravo,Yalda
AU  - Teriete,Peter
AU  - Dhanya,Raveendra-Panickar
AU  - Dahl,Russell
AU  - Lee,Pooi San
AU  - Kiffer-Moreira,Tina
AU  - Ganji,Santhi Reddy
AU  - Sergienko,Eduard
AU  - Smith,Layton H
AU  - Farquharson,Colin
AU  - Millán,José Luis
AU  - Cosford,Nicholas D P
TI  - Design, synthesis and evaluation of benzoisothiazolones as selective inhibitors of PHOSPHO1
SN  - 1464-3405
PY  - 2015///0330
KW  - Animals
KW  - Benzamides
KW  - chemical synthesis
KW  - Benzothiazoles
KW  - Dose-Response Relationship, Drug
KW  - Drug Design
KW  - Enzyme Inhibitors
KW  - Hepatocytes
KW  - drug effects
KW  - High-Throughput Screening Assays
KW  - Humans
KW  - Hydrogen-Ion Concentration
KW  - Mice
KW  - Molecular Structure
KW  - Phosphoric Monoester Hydrolases
KW  - antagonists & inhibitors
KW  - Small Molecule Libraries
KW  - Structure-Activity Relationship
N1  - Publication Type: Journal Article; Research Support, American Recovery and Reinvestment Act; Research Support, N.I.H., Extramural
UR  - https://doi.org/10.1016/j.bmcl.2014.07.013
ER  -