Bravo, Yalda

Design, synthesis and evaluation of benzoisothiazolones as selective inhibitors of PHOSPHO1. [electronic resource] - Bioorganic & medicinal chemistry letters Sep 2014 - 4308-11 p. digital

Publication Type: Journal Article; Research Support, American Recovery and Reinvestment Act; Research Support, N.I.H., Extramural

1464-3405

10.1016/j.bmcl.2014.07.013 doi


Animals
Benzamides--chemical synthesis
Benzothiazoles--chemical synthesis
Dose-Response Relationship, Drug
Drug Design
Enzyme Inhibitors--chemical synthesis
Hepatocytes--drug effects
High-Throughput Screening Assays
Humans
Hydrogen-Ion Concentration
Mice
Molecular Structure
Phosphoric Monoester Hydrolases--antagonists & inhibitors
Small Molecule Libraries--chemical synthesis
Structure-Activity Relationship