TY - GEN AU - Malherbe,Pari AU - Knoflach,Frédéric AU - Marcuz,Anne AU - Bohnert,Claudia AU - Weber,Michael AU - Knust,Henner AU - Ratni,Hasane AU - Spooren,Will AU - Ballard,Theresa M AU - Bissantz,Caterina TI - Mapping the binding pocket of a novel, high-affinity, slow dissociating tachykinin NK3 receptor antagonist: biochemical and electrophysiological characterization SN - 1873-7064 PY - 2015///0714 KW - Amino Acid Sequence KW - Animals KW - Antipsychotic Agents KW - pharmacology KW - Binding Sites KW - Carbamates KW - pharmacokinetics KW - Central Nervous System Agents KW - Dopaminergic Neurons KW - drug effects KW - Female KW - Gerbillinae KW - Guinea Pigs KW - HEK293 Cells KW - Humans KW - Locomotion KW - Male KW - Models, Molecular KW - Molecular Sequence Data KW - Mutation KW - Neurotransmitter Agents KW - Pars Compacta KW - Peptide Fragments KW - Piperidines KW - Receptors, Neurokinin-2 KW - antagonists & inhibitors KW - Receptors, Neurokinin-3 KW - agonists KW - Substance P KW - analogs & derivatives KW - Tissue Culture Techniques N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/j.neuropharm.2014.07.017 ER -