Malherbe, Pari
Mapping the binding pocket of a novel, high-affinity, slow dissociating tachykinin NK3 receptor antagonist: biochemical and electrophysiological characterization. [electronic resource]
- Neuropharmacology Nov 2014
- 259-72 p. digital
Publication Type: Journal Article
ISSN: 1873-7064
Standard No.: 10.1016/j.neuropharm.2014.07.017 doi
Subjects--Topical Terms: Amino Acid Sequence Animals Antipsychotic Agents--pharmacology Binding Sites Carbamates--pharmacokinetics Central Nervous System Agents--pharmacology Dopaminergic Neurons--drug effects Female Gerbillinae Guinea Pigs HEK293 Cells Humans Locomotion--drug effects Male Models, Molecular Molecular Sequence Data Mutation Neurotransmitter Agents--pharmacokinetics Pars Compacta--drug effects Peptide Fragments--pharmacology Piperidines--pharmacokinetics Receptors, Neurokinin-2--antagonists & inhibitors Receptors, Neurokinin-3--agonists Substance P--analogs & derivatives Tissue Culture Techniques