Li, Zhenyu

Design, synthesis and biological evaluation of 17-arylmethylamine-17-demethoxygeldanamycin derivatives as potent Hsp90 inhibitors. [electronic resource] - European journal of medicinal chemistry Oct 2014 - 359-70 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1768-3254

10.1016/j.ejmech.2014.07.101 doi


Animals
Antineoplastic Agents--chemical synthesis
Benzoquinones--chemical synthesis
Cell Line, Tumor
Cell Proliferation--drug effects
Chemistry Techniques, Synthetic
Drug Design
HSP90 Heat-Shock Proteins--antagonists & inhibitors
Humans
Lactams, Macrocyclic--chemical synthesis
Liver--drug effects
Male
Mice
Models, Molecular
Protein Conformation