Ma, Shao-lin

Lapatinib antagonizes multidrug resistance-associated protein 1-mediated multidrug resistance by inhibiting its transport function. [electronic resource] - Molecular medicine (Cambridge, Mass.) Sep 2014 - 390-9 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1528-3658

10.2119/molmed.2014.00059 doi


Animals
Antineoplastic Agents--pharmacology
Biological Transport--drug effects
Cell Line, Tumor
Cell Survival--drug effects
Cisplatin--pharmacology
Doxorubicin--pharmacology
Drug Resistance, Multiple--drug effects
Drug Resistance, Neoplasm--drug effects
Drug Synergism
Extracellular Signal-Regulated MAP Kinases--metabolism
HEK293 Cells
Humans
Lapatinib
Mice
Mice, Nude
Multidrug Resistance-Associated Protein 2
Multidrug Resistance-Associated Proteins--antagonists & inhibitors
NIH 3T3 Cells
Neoplasms--drug therapy
Proto-Oncogene Proteins c-akt--metabolism
Quinazolines--pharmacology
Tumor Burden--drug effects
Vincristine--pharmacology