TY - GEN AU - Takhi,Mohamed AU - Sreenivas,Kandepu AU - Reddy,Chandrashekar K AU - Munikumar,Mahadari AU - Praveena,Kolakota AU - Sudheer,Pabolu AU - Rao,Bandaru N V M AU - Ramakanth,Gollamudi AU - Sivaranjani,Jampala AU - Mulik,Shardaprasad AU - Reddy,Yeruva R AU - Narasimha Rao,Krishnamurthy AU - Pallavi,Rentala AU - Lakshminarasimhan,Anirudha AU - Panigrahi,Sunil K AU - Antony,Thomas AU - Abdullah,Iskandar AU - Lee,Yean K AU - Ramachandra,Murali AU - Yusof,Rohana AU - Rahman,Noorsaadah A AU - Subramanya,Hosahalli TI - Discovery of azetidine based ene-amides as potent bacterial enoyl ACP reductase (FabI) inhibitors SN - 1768-3254 PY - 2015///0417 KW - Amides KW - chemistry KW - Animals KW - Azetidines KW - Crystallography, X-Ray KW - Dose-Response Relationship, Drug KW - Drug Discovery KW - Enoyl-(Acyl-Carrier-Protein) Reductase (NADH) KW - metabolism KW - Enzyme Inhibitors KW - Male KW - Mice KW - Microsomes, Liver KW - Models, Molecular KW - Molecular Structure KW - Staphylococcus aureus KW - cytology KW - Structure-Activity Relationship N1 - Publication Type: Journal Article; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1016/j.ejmech.2014.07.036 ER -