Boucherle, Benjamin

A new 9-alkyladenine-cyclic methylglyoxal diadduct activates wt- and F508del-cystic fibrosis transmembrane conductance regulator (CFTR) in vitro and in vivo. [electronic resource] - European journal of medicinal chemistry Aug 2014 - 455-65 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1768-3254

10.1016/j.ejmech.2014.06.028 doi


Adenine--chemistry
Animals
CHO Cells
Cricetinae
Cricetulus
Cystic Fibrosis Transmembrane Conductance Regulator--chemistry
Drug Design
Humans
Male
Models, Molecular
Protein Conformation
Rats
Sequence Deletion