Boltjes, André

Fragment-based library generation for the discovery of a peptidomimetic p53-Mdm4 inhibitor. [electronic resource] - ACS combinatorial science Aug 2014 - 393-6 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

2156-8944

10.1021/co500026b doi


Drug Discovery
Humans
Ligands
Models, Molecular
Molecular Docking Simulation
Peptidomimetics--chemistry
Protein Interaction Maps--drug effects
Proto-Oncogene Proteins c-mdm2--antagonists & inhibitors
Tumor Suppressor Protein p53--antagonists & inhibitors