Fragment-based library generation for the discovery of a peptidomimetic p53-Mdm4 inhibitor. [electronic resource]
- ACS combinatorial science Aug 2014
- 393-6 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
2156-8944
10.1021/co500026b doi
Drug Discovery Humans Ligands Models, Molecular Molecular Docking Simulation Peptidomimetics--chemistry Protein Interaction Maps--drug effects Proto-Oncogene Proteins c-mdm2--antagonists & inhibitors Tumor Suppressor Protein p53--antagonists & inhibitors