TY  - GEN
AU  - Schoultz,Bent W
AU  - Hjørnevik,Trine
AU  - Reed,Brian J
AU  - Marton,János
AU  - Coello,Christopher S
AU  - Willoch,Frode
AU  - Henriksen,Gjermund
TI  - Synthesis and evaluation of three structurally related ¹⁸F-labeled orvinols of different intrinsic activities: 6-O-[¹⁸F]fluoroethyl-diprenorphine ([¹⁸F]FDPN), 6-O-[¹⁸F]fluoroethyl-buprenorphine ([¹⁸F]FBPN), and 6-O-[¹⁸F]fluoroethyl-phenethyl-orvinol ([¹⁸F]FPEO)
SN  - 1520-4804
PY  - 2014///0905
KW  - Animals
KW  - Brain
KW  - diagnostic imaging
KW  - Buprenorphine
KW  - analogs & derivatives
KW  - CHO Cells
KW  - Carbon Radioisotopes
KW  - Cricetulus
KW  - Diprenorphine
KW  - Fluorine Radioisotopes
KW  - Humans
KW  - Morphinans
KW  - chemical synthesis
KW  - Narcotic Antagonists
KW  - Positron-Emission Tomography
KW  - Radioligand Assay
KW  - Radiopharmaceuticals
KW  - Rats
KW  - Receptors, Opioid
KW  - agonists
KW  - Structure-Activity Relationship
N1  - Publication Type: Journal Article
UR  - https://doi.org/10.1021/jm500503k
ER  -