TY - GEN AU - Abdelsamie,Ahmed S AU - Bey,Emmanuel AU - Hanke,Nina AU - Empting,Martin AU - Hartmann,Rolf W AU - Frotscher,Martin TI - Inhibition of 17β-HSD1: SAR of bicyclic substituted hydroxyphenylmethanones and discovery of new potent inhibitors with thioether linker SN - 1768-3254 PY - 2015///0330 KW - 17-Hydroxysteroid Dehydrogenases KW - antagonists & inhibitors KW - Animals KW - Dose-Response Relationship, Drug KW - Drug Discovery KW - Enzyme Inhibitors KW - chemical synthesis KW - Humans KW - Mice KW - Models, Molecular KW - Molecular Structure KW - Phenols KW - Structure-Activity Relationship KW - Sulfides KW - chemistry N1 - Publication Type: Journal Article; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1016/j.ejmech.2014.05.074 ER -