Johnson, James A

Design, synthesis and evaluation of phenethylaminoheterocycles as K(v)1.5 inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Jul 2014 - 3018-22 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2014.05.035 doi


Animals
Carbamates--chemical synthesis
Dose-Response Relationship, Drug
Drug Design
Heart Atria--drug effects
Heart Rate--drug effects
Humans
Indazoles--chemical synthesis
Kv1.5 Potassium Channel--antagonists & inhibitors
Models, Molecular
Molecular Structure
Potassium Channel Blockers--chemical synthesis
Rabbits
Rats
Structure-Activity Relationship