Parkkari, Teija

Discovery of triterpenoids as reversible inhibitors of α/β-hydrolase domain containing 12 (ABHD12). [electronic resource] - PloS one 2014 - e98286 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1932-6203

10.1371/journal.pone.0098286 doi


Animals
Drug Discovery
Enzyme Inhibitors--chemistry
HEK293 Cells
Humans
Ligands
Mice
Molecular Docking Simulation
Monoacylglycerol Lipases--antagonists & inhibitors
Protein Conformation
Structure-Activity Relationship
Substrate Specificity
Triterpenes--chemistry