Appleton, Kathryn M
Development of inhibitors of heterotrimeric Gαi subunits. [electronic resource]
- Bioorganic & medicinal chemistry Jul 2014
- 3423-34 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1464-3391
10.1016/j.bmc.2014.04.035 doi
Cells, Cultured
Dose-Response Relationship, Drug
Drug Discovery
GTP-Binding Protein alpha Subunits, Gi-Go--antagonists & inhibitors
HEK293 Cells
Humans
Models, Molecular
Molecular Structure
Peptides--chemical synthesis
Small Molecule Libraries--chemistry
Structure-Activity Relationship