Appleton, Kathryn M

Development of inhibitors of heterotrimeric Gαi subunits. [electronic resource] - Bioorganic & medicinal chemistry Jul 2014 - 3423-34 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1464-3391

10.1016/j.bmc.2014.04.035 doi


Cells, Cultured
Dose-Response Relationship, Drug
Drug Discovery
GTP-Binding Protein alpha Subunits, Gi-Go--antagonists & inhibitors
HEK293 Cells
Humans
Models, Molecular
Molecular Structure
Peptides--chemical synthesis
Small Molecule Libraries--chemistry
Structure-Activity Relationship