Graham, Thomas H

Pyrazoles as non-classical bioisosteres in prolylcarboxypeptidase (PrCP) inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Apr 2014 - 1657-60 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2014.02.070 doi


Animals
Carboxypeptidases--antagonists & inhibitors
Dose-Response Relationship, Drug
Enzyme Inhibitors--chemical synthesis
Humans
Mice
Molecular Structure
Pyrazoles--chemical synthesis
Structure-Activity Relationship