Graham, Thomas H
Pyrazoles as non-classical bioisosteres in prolylcarboxypeptidase (PrCP) inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry letters Apr 2014
- 1657-60 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2014.02.070 doi
Animals
Carboxypeptidases--antagonists & inhibitors
Dose-Response Relationship, Drug
Enzyme Inhibitors--chemical synthesis
Humans
Mice
Molecular Structure
Pyrazoles--chemical synthesis
Structure-Activity Relationship