Cyclic marinopyrrole derivatives as disruptors of Mcl-1 and Bcl-x(L) binding to Bim. [electronic resource]
- Marine drugs Mar 2014
- 1335-48 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1660-3397
10.3390/md12031335 doi
Apoptosis--drug effects Apoptosis Regulatory Proteins--chemistry Bcl-2-Like Protein 11 Blotting, Western Breast Neoplasms--drug therapy Catalysis Cell Line, Tumor Drug Screening Assays, Antitumor Enzyme-Linked Immunosorbent Assay Female Humans Indicators and Reagents Isomerism Magnetic Resonance Spectroscopy Marine Toxins--pharmacology Membrane Proteins--chemistry Myeloid Cell Leukemia Sequence 1 Protein--metabolism Protein Binding--drug effects Proto-Oncogene Proteins--chemistry Pyrroles--chemical synthesis Spectrophotometry, Ultraviolet Structure-Activity Relationship bcl-X Protein--metabolism