Megens, Anton A H P

Pharmacology of JNJ-42314415, a centrally active phosphodiesterase 10A (PDE10A) inhibitor: a comparison of PDE10A inhibitors with D2 receptor blockers as potential antipsychotic drugs. [electronic resource] - The Journal of pharmacology and experimental therapeutics Apr 2014 - 138-54 p. digital

Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't

1521-0103

10.1124/jpet.113.211904 doi


Animals
Antipsychotic Agents--chemistry
Behavior, Animal--drug effects
Brain--drug effects
Dopamine Antagonists--chemistry
Dopamine D2 Receptor Antagonists
Female
Guinea Pigs
Humans
Imidazoles--pharmacology
Male
Motor Activity--drug effects
Phosphodiesterase Inhibitors--chemistry
Phosphoric Diester Hydrolases--genetics
Prolactin--metabolism
Protein Binding
Pyrazines--pharmacology
Rats
Rats, Inbred Lew
Rats, Sprague-Dawley
Rats, Wistar
Sf9 Cells
Spodoptera
Stereotyped Behavior--drug effects