Caglič, Dejan

Identification of clinically viable quinolinol inhibitors of botulinum neurotoxin A light chain. [electronic resource] - Journal of medicinal chemistry Feb 2014 - 669-76 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1520-4804

10.1021/jm4012164 doi


Animals
Botulinum Toxins, Type A--antagonists & inhibitors
Catalytic Domain
Humans
Hydrogen-Ion Concentration
Hydroxyquinolines--chemical synthesis
In Vitro Techniques
Microsomes, Liver--metabolism
Rats
Rats, Sprague-Dawley
Solubility
Structure-Activity Relationship