Thurner, Patrick

Mechanism of hERG channel block by the psychoactive indole alkaloid ibogaine. [electronic resource] - The Journal of pharmacology and experimental therapeutics Feb 2014 - 346-58 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1521-0103

10.1124/jpet.113.209643 doi


Amino Acid Substitution
Binding Sites--drug effects
Cell Line
Cytosol--metabolism
ERG1 Potassium Channel
Ether-A-Go-Go Potassium Channels--antagonists & inhibitors
Excitatory Amino Acid Antagonists--adverse effects
Hallucinogens--adverse effects
Humans
Hydrogen-Ion Concentration
Ibogaine--adverse effects
Ion Channel Gating--drug effects
Kinetics
Membrane Potentials--drug effects
Membrane Transport Modulators--pharmacology
Molecular Conformation
Molecular Docking Simulation
Mutant Proteins--agonists
Narcotic Antagonists--adverse effects
Nerve Tissue Proteins--antagonists & inhibitors
Recombinant Proteins--chemistry