N-(3-(2-amino-6,6-difluoro-4,4a,5,6,7,7a-hexahydro-cyclopenta[e][1,3]oxazin-4-yl)-phenyl)-amides as BACE1 inhibitors: a patent evaluation of WO2013041499. [electronic resource]
- Expert opinion on therapeutic patents Feb 2014
- 239-42 p. digital
Publication Type: Journal Article; Review
1744-7674
10.1517/13543776.2014.859246 doi
Alzheimer Disease--drug therapy Amides--chemistry Amyloid Precursor Protein Secretases--antagonists & inhibitors Amyloid beta-Protein Precursor--metabolism Animals Aspartic Acid Endopeptidases--antagonists & inhibitors Drug Design Drug and Narcotic Control Humans Molecular Structure Molecular Targeted Therapy Oxazines--chemistry Patents as Topic Protease Inhibitors--chemistry Structure-Activity Relationship