Dessolin, Jean

N-(3-(2-amino-6,6-difluoro-4,4a,5,6,7,7a-hexahydro-cyclopenta[e][1,3]oxazin-4-yl)-phenyl)-amides as BACE1 inhibitors: a patent evaluation of WO2013041499. [electronic resource] - Expert opinion on therapeutic patents Feb 2014 - 239-42 p. digital

Publication Type: Journal Article; Review

1744-7674

10.1517/13543776.2014.859246 doi


Alzheimer Disease--drug therapy
Amides--chemistry
Amyloid Precursor Protein Secretases--antagonists & inhibitors
Amyloid beta-Protein Precursor--metabolism
Animals
Aspartic Acid Endopeptidases--antagonists & inhibitors
Drug Design
Drug and Narcotic Control
Humans
Molecular Structure
Molecular Targeted Therapy
Oxazines--chemistry
Patents as Topic
Protease Inhibitors--chemistry
Structure-Activity Relationship