Bin, Jin Wen

Structure-activity relationship study of permethyl ningalin B analogues as P-glycoprotein chemosensitizers. [electronic resource] - Journal of medicinal chemistry Nov 2013 - 9057-70 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/jm400930e doi


ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism
ATP Binding Cassette Transporter, Subfamily G, Member 2
ATP-Binding Cassette Transporters--metabolism
Cell Line, Tumor
Doxorubicin--metabolism
Drug Resistance, Neoplasm--drug effects
Heterocyclic Compounds, 3-Ring--chemistry
Humans
Intracellular Space--drug effects
Models, Molecular
Molecular Conformation
Multidrug Resistance-Associated Proteins--metabolism
Neoplasm Proteins--metabolism
Paclitaxel--pharmacology
Safety
Structure-Activity Relationship