Feng, Taotao

The discovery of novel histone lysine methyltransferase G9a inhibitors (part 1): molecular design based on a series of substituted 2,4-diamino-7- aminoalkoxyquinazoline by molecular-docking-guided 3D quantitative structure-activity relationship studies. [electronic resource] - Medicinal chemistry (Shariqah (United Arab Emirates)) Jun 2014 - 426-40 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1875-6638

10.2174/15734064113096660068 doi


Dose-Response Relationship, Drug
Drug Discovery
Enzyme Inhibitors--chemical synthesis
Histone-Lysine N-Methyltransferase--antagonists & inhibitors
Humans
Molecular Docking Simulation
Molecular Structure
Quantitative Structure-Activity Relationship
Quinazolines--chemical synthesis