Na+/H+ exchanger 1 is regulated via its lipid-interacting domain, which functions as a molecular switch: a pharmacological approach using indolocarbazole compounds. [electronic resource]
- Molecular pharmacology Jan 2014
- 18-28 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1521-0111
10.1124/mol.113.089268 doi
Adrenergic alpha-1 Receptor Agonists--pharmacology Animals Binding, Competitive Carbazoles--chemistry Cation Transport Proteins--antagonists & inhibitors Cell Membrane Cricetinae Cricetulus Databases, Chemical Indoles--chemistry Lipids--chemistry Maleimides--chemistry Mice Mutation Okadaic Acid--pharmacology Osmotic Pressure Phosphatidylinositol 4,5-Diphosphate--pharmacology Protein Kinase C--antagonists & inhibitors Protein Kinase Inhibitors--chemistry Protein Structure, Tertiary Protein Transport Receptors, Adrenergic, alpha-1--genetics Sodium-Hydrogen Exchanger 1 Sodium-Hydrogen Exchangers--antagonists & inhibitors Staurosporine--chemistry Transfection