Thiazolopyridine ureas as novel antitubercular agents acting through inhibition of DNA Gyrase B. [electronic resource]
- Journal of medicinal chemistry Nov 2013
- 8834-48 p. digital
Publication Type: Journal Article
1520-4804
10.1021/jm401268f doi
Animals Antitubercular Agents--administration & dosage DNA Gyrase--metabolism Disease Models, Animal Dose-Response Relationship, Drug Mice Mice, Inbred BALB C Models, Molecular Molecular Structure Mycobacterium tuberculosis--drug effects Pyridines--administration & dosage Structure-Activity Relationship Topoisomerase II Inhibitors--administration & dosage Tuberculosis--drug therapy Urea--analogs & derivatives