bba, a synthetic derivative of 23-hydroxybutulinic acid, reverses multidrug resistance by inhibiting the efflux activity of MRP7 (ABCC10). [electronic resource]
- PloS one 2013
- e74573 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1932-6203
10.1371/journal.pone.0074573 doi
ATP Binding Cassette Transporter, Subfamily B ATP Binding Cassette Transporter, Subfamily B, Member 1--genetics Adenosine Triphosphate--metabolism Antineoplastic Agents--metabolism Cell Line, Tumor Drug Resistance, Multiple--genetics Drug Resistance, Neoplasm Gene Expression HEK293 Cells Humans Inhibitory Concentration 50 Multidrug Resistance-Associated Proteins--antagonists & inhibitors Paclitaxel--metabolism Pentacyclic Triterpenes Protein Transport--drug effects Triterpenes--chemistry Betulinic Acid