TY - GEN AU - Perspicace,Enrico AU - Giorgio,Annalaura AU - Carotti,Angelo AU - Marchais-Oberwinkler,Sandrine AU - Hartmann,Rolf W TI - Novel N-methylsulfonamide and retro-N-methylsulfonamide derivatives as 17β-hydroxysteroid dehydrogenase type 2 (17β-HSD2) inhibitors with good ADME-related physicochemical parameters SN - 1768-3254 PY - 2014///0708 KW - Chemistry, Physical KW - Dose-Response Relationship, Drug KW - Enzyme Inhibitors KW - chemistry KW - Estradiol Dehydrogenases KW - antagonists & inhibitors KW - Humans KW - Molecular Structure KW - Structure-Activity Relationship KW - Sulfonamides KW - chemical synthesis N1 - Publication Type: Journal Article; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1016/j.ejmech.2013.08.026 ER -