Novel synthetic curcumin analogues EF31 and UBS109 are potent DNA hypomethylating agents in pancreatic cancer. [electronic resource]
- Cancer letters Dec 2013
- 195-203 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1872-7980
10.1016/j.canlet.2013.08.002 doi
Animals Blotting, Western Cadherins--genetics Cell Line, Tumor Cell Proliferation--drug effects Cell Survival--drug effects Curcumin--analogs & derivatives Cytosine--metabolism DNA (Cytosine-5-)-Methyltransferase 1 DNA (Cytosine-5-)-Methyltransferases--genetics DNA Methylation--drug effects Dose-Response Relationship, Drug Female Gene Expression Regulation, Neoplastic--drug effects HSP90 Heat-Shock Proteins--genetics Humans Immunohistochemistry Mice Mice, Nude Osteonectin--genetics Pancreatic Neoplasms--drug therapy Piperidones--pharmacology Pyridines Reverse Transcriptase Polymerase Chain Reaction Xenograft Model Antitumor Assays